Site Specific Linkers
Site-Specific linkers offer precise coupling of cytotoxins or chemotherapeutic drugs to specific sites within antibody molecules. They ensure ADCs exhibit high homogeneity and an increased therapeutic index (TI). Beyond traditional cytotoxin-conjugated ADCs, site-specific linkers facilitate the development of various immunoconjugates, promising enhanced efficacy and safety across a broad spectrum of challenging diseases.
- Mono-Sulfone Acid
- Sulfone-PEG-Acid
- Mono-Sulfone NHS Ester
- Sulfone-PEG-NHS ester
- Bis-sulfone Amine
- Bis-sulfone-PEG-Azide
- Bis-sulfone-PEG-Bis-sulfone
- Dibromo-Maleimide
- 3,4-Dibromo-Mal-PEG-Acid
- 3,4-Dibromo-Mal-PEG-NHS ester
- 3,4-Dibromo-Mal-PEG-t-butyl ester
- 3,4-Dibromo-Mal-PEG-Amine
- 3,4-Dibromo-Mal-PEG-Boc
- 3,4-Dibromo-Mal-PEG-Azide
- 3,4-Dibromo-Mal-PEG-DBCO
- 3,4-Dibromo-Mal-PEG-Methyltetrazine
- 3,4-Dibromo-Mal-PEG-Val-Cit-PAB-MMAE
- Biotin-PEG-3,4-Dibromo-Mal
- Diphenylthiol-Mal-PEG-Biotin
- Dithiophenol-Maleimide
Catalog | Product Name | Structure | M.W. | Purity | Pricing |
---|---|---|---|---|---|
Mono-Sulfone Acid | |||||
BP-40315 | Mono-Sulfone Acid | ![]() | 332.4 | Pricing | |
Sulfone-PEG-Acid | |||||
BP-22307 | 4-(3-tosyl-2-(tosylmethyl)propanoyl)benzoic acid | ![]() | 500.6 | 98% | Pricing |
BP-25492 | Bis-sulfone-PEG4-Acid | ![]() | 747.9 | 98% | Pricing |
BP-24476 | Bis-Sulfone-PEG8-acid | ![]() | 924.1 | 98% | Pricing |
BP-25619 | Bis-sulfone-PEG12-Acid | ![]() | 1100.3 | 98% | Pricing |
BP-23334 | Active-Mono-Sulfone-PEG8-acid | ![]() | 767.9 | 95% | Pricing |
Mono-Sulfone NHS Ester | |||||
BP-40316 | Mono-Sulfone NHS Ester | ![]() | 429.5 | Pricing | |
Sulfone-PEG-NHS ester | |||||
BP-23344 | Bis-sulfone NHS Ester | ![]() | 597.7 | 90% | Pricing |
BP-23343 | Bis-sulfone-PEG4-NHS Ester | ![]() | 845 | 93% | Pricing |
BP-23417 | Bis-sulfone-PEG8-NHS Ester | ![]() | 1021.2 | 95% | Pricing |
BP-23342 | Bis-sulfone-PEG12-NHS Ester | ![]() | 1197.4 | 90% | Pricing |
Bis-sulfone Amine | |||||
BP-40283 | Bis-sulfone Amine | ![]() | 556.7 | Pricing | |
Bis-sulfone-PEG-Azide | |||||
BP-40218 | Bis-sulfone-PEG4-azide | ![]() | 744.9 | 98% | Pricing |
BP-43519 | Bis-sulfone-PEG8-azide | ![]() | 921.1 | 98% | Pricing |
Bis-sulfone-PEG-Bis-sulfone | |||||
BP-41039 | Bis-sulfone-PEG1-Bis-sulfone | ![]() | 1069.3 | 95% | Pricing |
BP-41130 | Bis-sulfone-PEG2-Bis-sulfone | ![]() | 1113.4 | 95% | Pricing |
Dibromo-Maleimide | |||||
BP-23379 | 3,4-Dibromo-1H-pyrrole-2,5-dione | ![]() | 254.9 | Pricing | |
BP-21984 | methyl 3,4-dibromo-2,5-dioxo-2H-pyrrole-1(5H)-carboxylate | ![]() | 312.9 | 96% | Pricing |
BP-24171 | ethyl 3,4-dibromo-2,5-dioxo-2H-pyrrole-1(5H)-carboxylate | ![]() | 326.9 | 96% | Pricing |
3,4-Dibromo-Mal-PEG-Acid | |||||
BP-28207 | 3,4-Dibromo-Mal-PEG4-Acid | ![]() | 503.1 | Pricing | |
BP-23413 | 3,4-Dibromo-Mal-PEG8-acid | ![]() | 679.4 | 98% | Pricing |
3,4-Dibromo-Mal-PEG-NHS ester | |||||
BP-28208 | 3,4-Dibromo-Mal-PEG4-NHS ester | ![]() | 600.2 | Pricing | |
3,4-Dibromo-Mal-PEG-t-butyl ester | |||||
BP-23382 | 3,4-Dibromo-Mal-PEG4-t-butyl ester | ![]() | 559.3 | 98% | Pricing |
BP-23398 | 3,4-Dibromo-Mal-PEG8-t-butyl ester | ![]() | 735.5 | 98% | Pricing |
3,4-Dibromo-Mal-PEG-Amine | |||||
BP-22011 | 3,4-Dibromo-Mal-PEG2-Amine TFA salt | ![]() | 386 | 98% | Pricing |
BP-28209 | 3,4-Dibromo-Mal-PEG4-Amine | ![]() | 474.1 | Pricing | |
BP-28210 | 3,4-Dibromo-Mal-PEG8-Amine | ![]() | 650.4 | Pricing | |
3,4-Dibromo-Mal-PEG-Boc | |||||
BP-22016 | 3,4-Dibromo-Mal-PEG2-Boc-Amine | ![]() | 486.2 | 98% | Pricing |
BP-41739 | 3,4-Dibromo-Mal-PEG8-Boc-Amine | ![]() | 750.5 | 98% | Pricing |
3,4-Dibromo-Mal-PEG-Azide | |||||
BP-40217 | 3,4-Dibromo-Mal-PEG8-Azide | ![]() | 676.4 | 98% | Pricing |
3,4-Dibromo-Mal-PEG-DBCO | |||||
BP-29795 | 3,4-Dibromo-Mal-PEG4-amide-DBCO | ![]() | 761.5 | 98% | Pricing |
3,4-Dibromo-Mal-PEG-Methyltetrazine | |||||
BP-29734 | Methyltetrazine-PEG4-Amido-PEG8-Mal-3,4-Dibromo | ![]() | 1024.8 | 98% | Pricing |
3,4-Dibromo-Mal-PEG-Val-Cit-PAB-MMAE | |||||
BP-41473 | 3,4-Dibromo-Mal-PEG4-Val-Cit-PAB-MMAE | ![]() | 1608.6 | Pricing | |
BP-43740 | 3,4-Dibromo-Mal-PEG8-Val-Cit-PAB-MMAE | ![]() | 1784.8 | 97% | Pricing |
Biotin-PEG-3,4-Dibromo-Mal | |||||
BP-40277 | Biotin-PEG4-Amide-PEG8-3,4-Dibromo-Mal | ![]() | 1124 | 98% | Pricing |
Diphenylthiol-Mal-PEG-Biotin | |||||
BP-29550 | Diphenylthiol-Mal-PEG8-PEG4-Biotin | ![]() | 1182.5 | Pricing | |
Dithiophenol-Maleimide | |||||
BP-26116 | N-(Methyltetrazine-PEG4)-amido-PEG8-3,4-dithiophenolmaleimide | ![]() | 1083.3 | Pricing |