6-((2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)-N-(4-(6-methyl-1,2,4,5-tetrazin-3-yl)benzyl)hexanamide

6-((2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)-N-(4-(6-methyl-1,2,4,5-tetrazin-3-yl)benzyl)hexanamide


6-((2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)-N-(4-(6-methyl-1,2,4,5-tetrazin-3-yl)benzyl)hexanamide is a PROTAC linker featuring a thalidomide, a hydrophilic PEG spacer, and a methyltetrazine. Thalidomide is a ligand for E3 ligase, which marks proteins for proteolysis. Meanwhile, the methyltetrazine is a click chemistry handle used to form bonds with TCO groups on target molecules.

Molecular structure of the compound BP-40569
    • Unit
    • Price
    • Qty
    • 50 MG
    • $450.00
    • 100 MG
    • $850.00

Usually ships within 24 hours.


Would you like to inquire about custom quantity?
Inquire