RVX-208

RVX-208


Apabetalone (RVX-208) is an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain. Apabetalone has C50s are 87+/-10 μM and 0.51+/-0.041 μM for BD1 and BD2, respectively. Apabetalone binds to the acetyl-lysine binding pocket in a peptide-competitive way, which accounts for its pharmacological activity. Reagent grade, for research purpose. Please contact us for GMP-grade inquiries.

Molecular structure of the compound BP-23380
    • Unit
    • Price
    • Qty
    • 10 MG
    • $280.00
    • 25 MG
    • $490.00
    • 50 MG
    • $780.00

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